阿拉丁小分子抑制劑、激動劑、拮抗劑--DNA損傷/DNA修復信號通路-商家動態-資訊-生物在線

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阿拉丁小分子抑制劑、激動劑、拮抗劑--DNA損傷/DNA修復信號通路

作者:上海阿拉丁生化科技股份有限公司 2020-11-27T09:22 (訪問量:6517)

">K126884KU-55933 (ATM Kinase Inhibitor)≥98%587871-26-95mg,25mg,100mg無細胞ATM12.9 nM2.2 nMK127121KU-60019≥98%925701-49-15mg,25mg,100mg無細胞ATM6.3 nMV125220VE-821≥98%1232410-49-95mg,25mg,100mg無細胞ATR13 nM26 nMW100984Wortmannin98%19545-26-75mg,10mg,25mg無細胞PI3K3 nMDNA-PK/ATM16 nMDNA-PK/ATM150 nMT129646Torin 2≥98%1223001-51-15mg,10mg,50mgp53?/? MEFs細胞系mTOR0.25 nMPC3細胞系ATM/ATR/DNA-PK 28 nMATM/ATR/DNA-PK 35 nMATM/ATR/DNA-PK 118 nMC128014CP-466722≥98%1080622-86-15mg,25mgATM410 nME125288ETP-46464≥99%1345675-02-610mg,50mgATR25 nMC129735CGK 733≥99%905973-89-95mg,10mg,50mgATM200 nMATR200 nMA125603AZ20≥98%1233339-22-45mg,10mg,50mg無細胞ATR5 nMS117968五味子乙素分析標準品,>98%61281-37-625mg,100mgATR7.25 μMC129284磷酸氯喹≥99%50-63-55g,10g,25g,100g,500g ATM

*PARP

項目號產品名稱規格CAS包裝細胞靶點IC50KiEC50
O126162Olaparib (AZD2281, Ku-0059436)≥98%763113-22-010mg,25mg,100mg,250mg,1g,5gPARP15 nM
PARP21 nM
V127105Veliparib≥99%912444-00-910mg,50mg,250mg無細胞PARP15.2 nM
PARP22.9 nM
R129879Rucaparib (AG-014699,PF-01367338)≥99%459868-92-95mg,10mg,50mg PARP1.4 nM
B125751Iniparib (BSI-201)≥98%160003-66-710mg,50mg,250mg
B127705BMN 673≥98%1207456-01-610mg,50mg
A125467AG14361≥98%328543-09-55mg,10mg,50mg無細胞PARP1<5 nM
A1072073-氨基苯甲酰胺98%3544-24-91g,5g,25g,100gCHO細胞PARP<50 nM
P129886PJ34 HCl≥97%344458-15-75mg,25mg,100mg PARP 20 nM
M127627MK-4827 (Niraparib)98%1038915-60-410mg,50mg,100mgPARP1 3.8 nM
PARP22.1 nM
U129885UPF 1069≥98%1048371-03-410mg,50mgPARP18.0 μM
PARP20.3 μM
A127274AZD2461≥98%1174043-16-35mg,25mg,100mg PARP
H1571724-羥基喹唑啉≥98.0%(HPLC)491-36-15g,25g,100g
B110551苯甲酰胺99%55-21-025g,100g,500g,2.5kg PARP3.3 μM
B110552苯甲酰胺AR,98%55-21-025g,100g,500g PARP3.3 μM
B118608苯甲酰胺99.5%,升華純化55-21-05g,25gPARP3.3 μM
P138238吡啶酰胺≥98.0%(HPLC)1452-77-35g,25g,100g PARP95 μM  

*DNA/RNA合成

    項目號產品名稱規格CAS包裝細胞靶點IC50KiKd
    G120180鹽酸吉西他濱98%122111-03-910mg,50mg,250mg,1g,5g,25gPANC1細胞DNA合成50 nM
    MIAPaCa2細胞40 nM
    BxPC3細胞18 nM
    Capan2細胞12 nM
    P129841Pemetrexed≥99%150399-23-850mg,250mg無細胞TS1.3 nM
    DHFR7.2 nM
    GARFT65 nM
    C110682卡鉑98%41575-94-4100mg,250mg,1g,5g
    P124220噴司他丁98%(HPLC)53910-25-15mg,25mg
    F122998氟達拉濱98%21679-14-150mg,250mg,1g,5g
    O124003奧沙利鉑99%61825-94-325mg,100mg,500mg
    C127663CX-5461≥98%1138549-36-65mg,25mg,100mgHCT-116細胞rRNA合成142 nM
    A375細胞
    MIA PaCa-2細胞
    F1001495-氟尿嘧啶99%51-21-81g,5g,25g,100g,500g
    C124969Capecitabine≥99%154361-50-9250mg,1g,5g,25g
    F122999單磷酸氟達拉濱99%75607-67-925mg,100mg,500mg
    C126447Cidofovir≥98%113852-37-225mg,100mg
    C111218阿糖胞苷98%147-94-41g,5g,25g,100g
    G127944Gemcitabine≥99%95058-81-450mg,100mg,250mg,1g,5g,25g
    D129529Daptomycin≥98%103060-53-310mg,50mg,100mg,1g
    C129833Cladribine≥98%4291-63-810mg,50mg,100mg,250mg,25gU266, RPMI8226MM1.S細胞腺苷脫氨酶2.43 μM
    U266, RPMI8226MM1.S細胞0.75 μM
    U266, RPMI8226MM1.S細胞0.18 μM
    R129835Raltitrexed≥98%112887-68-010mg,50mg,100mg
    C102625克羅拉濱99%123318-82-15mg,20mg,25mg,100mg,500mg Ribonucleotide reductase65 nM
    I123381異環磷酰胺藥用級3778-73-250mg,250mg,1g,5g
    I123242異環磷酰胺98%3778-73-21g,5g,25g
    N129848NSC 207895≥99%58131-57-01mg,5mg,10mg,50mg MDMX2.5 μM
    D129847Dacarbazine≥98%4342-03-41g,5g,25g
    H106352羥基脲98%127-07-11g,5g,25g,100g
    F1107325-氟-2'-脫氧尿苷99%50-91-9100mg,250mg,500mg,1g,5g,25g
    M1268586-巰基嘌呤 (6-MP)≥99%50-44-250mg,250mg,1g,5g,25g,100g
    M129842Mizoribine≥98%50924-49-710mg,50mg,100mg,250mg
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